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P2X and P2Y Receptors Mediate Contraction Induced by Electrical Field Stimulation in Feline Esophageal Smooth Muscle
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  • P2X and P2Y Receptors Mediate Contraction Induced by Electrical Field Stimulation in Feline Esophageal Smooth Muscle
저자명
YoungRaeCho,HyeonSoonJang,WonKim,SunYoungPark,UyDongSohn
간행물명
The Korean Journal of Physiology & PharmacologyKCI,SCI,SCOPUS
권/호정보
2010년|14권 5호(통권83호)|pp.311-316 (6 pages)
발행정보
대한생리학회-대한약리학회|한국
파일정보
정기간행물|ENG|
PDF텍스트(4.12MB)
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영문초록

It is well-known that electrical field stimulation (EFS)-induced contraction is mediated by a cholinergic mechanism and other neurotransmitters. NO, ATP, calcitonin gene-related peptide (CGRP), and substance P are released by EFS. To investigate the purinergic mechanism involved in the EFS-induced contraction, purinegic receptors antagonists were used. Suramine, a non-selective P2 receptor antagonist, reduced the contraction induced by EFS. NF023 (10−7∼10−4 M), a selective P2X antagonist, inhibited the contraction evoked by EFS. Reactive blue (10−6∼10−4 M), selective P2Y antagonist, also blocked the contraction in a dose-dependent manner. In addition, P2X agonist Ձ,Ղ-methylene 5'-adenosine triphosphate (ՁՂMeATP, 10−7∼10−5 M) potentiated EFS-induced contrac</SUP>tion in a dose-dependent manner. P2Y agonist adenosine 5'-[Ղ-thio]diphosphate trilithium salt (ADPՂS, 10−7∼10−5 M) also potentiated EFS-induced contractions in a dose-dependent manner. Ecto-ATPase activator apyrase (5 and 10 U/ml) reduced EFS-induced contractions. Inversely, 6-N,N-diethyl-D-Ղ,Ճ- dibromomethylene 5'-triphosphate triammonium (ARL 67156, 10−4 M) increased EFS-induced contraction. These data suggest that endogenous ATP plays a role in EFS-induced contractions which are mediated through both P2X-receptors and P2Y-receptors stimulation in cat esophageal smooth muscle.

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